• Medientyp: E-Artikel
  • Titel: Discovery of Trifluoromethyl(pyrimidin-2-yl)azetidine-2-carboxamides as Potent, Orally Bioavailable TGR5 (GPBAR1) Agonists: Structure–Activity Relationships, Lead Optimization, and Chronic In Vivo Efficacy
  • Beteiligte: Phillips, Dean P.; Gao, Wenqi; Yang, Yang; Zhang, Guobao; Lerario, Isabelle K.; Lau, Thomas L.; Jiang, Jiqing; Wang, Xia; Nguyen, Deborah G.; Bhat, B. Ganesh; Trotter, Carol; Sullivan, Heather; Welzel, Gustav; Landry, Jannine; Chen, Yali; Joseph, Sean B.; Li, Chun; Gordon, W. Perry; Richmond, Wendy; Johnson, Kevin; Bretz, Angela; Bursulaya, Badry; Pan, Shifeng; McNamara, Peter;
  • Erschienen: American Chemical Society (ACS), 2014
  • Erschienen in: Journal of Medicinal Chemistry
  • Sprache: Englisch
  • DOI: 10.1021/jm401731q
  • ISSN: 0022-2623; 1520-4804
  • Entstehung:
  • Anmerkungen: